PBIT

• Description:

  PBIT inhibits JARID1B histone demethylase (IC50 of about 3 μM) . PBIT also inhibits JARID1A and JARID1C (IC50s of 6 μM and 4.9 μM, respectively) . PBIT is a specific inhibitor of the Jumonji AT-rich Interactive Domain 1 (JARID1) enzymes . PBIT, which inhibits JARID1B with an IC50 of about 3 μm in vitro.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  241.31

• Molecular Formula:

  C14H11NOS

• Notes:

  Research use only, not for human use.

• Receptor:

  JARID1B|JARID1A|JARID1C

• CAS Number:

  2514-30-9