KRM-II-81

• Description:

  KRM-II-81 is a potent, selective α1/α2/α3 GABAA receptors positive allosteric modulator with EC50 of 937 nM for α1β3γ2, negligible efficacy at α4/α5/α6 GABAA receptors.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  351.369

• Molecular Formula:

  C21H13N5O

• Notes:

  Research use only, not for human use.

• Receptor:

  GAT

• CAS Number:

  2014348-91-3