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Gavestinel

CAT: 0804-HY-150138-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-150138-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Gavestinel (GV 150526) is a selective and potent the glycine site of the NMDA receptor antagonist. Gavestinel has neuroprotectant effects[1].
CAS Number
153436-22-7
Product Name Alternative
GV 150526
UNSPSC
12352005
Target
IGluR
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
Neuroscience-Neurodegeneration
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/gavestinel.html
Purity
98.74
Solubility
DMSO : 125 mg/mL (ultrasonic)
Smiles
O=C(C(N1)=C(/C=C/C(NC2=CC=CC=C2)=O)C3=C1C=C(Cl)C=C3Cl)O
Molecular Formula
C18H12Cl2N2O3
Molecular Weight
375.21
References & Citations
[1]J F Hoke, et al. Pharmacokinetics of a glycine site antagonist (gavestinel) following multiple dosing in patients with acute stroke. Eur J Clin Pharmacol. 2000 Feb-Mar;55 (11-12) :867-72.
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, protect from light)
Scientific Category
Reference compound1
Clinical Information
Phase 2