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BI-9564

CAT: 0421-82064Size: 25 mgDry Ice: NoHazardous: No
CAT#:0421-82064Size:25 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
BI-9564 inhibits BRD9 and BRD7 bromodomains and exhibits no significant off-target pharmacology against a panel of 324 kinases and 55 GPCRs at concentrations less than 5 μM. BI-9564 is a selective inhibitor of BRD9 and BRD7 bromodomains (Kds = 14.1 and 239 nM; IC50s = 75 nM and 3.4 μM, respectively) that demonstrates cellular activity by semi-quantitative FRAP assay with ~90% inhibition of BRD9 and BRD7 at 0.1 μM and 1 μM, respectively. Inhibits proliferation of AML cell lines in vitro and reduces AML tumor xenograft growth in vivo.
CAS Number
1883429-22-8
Format
Solid
Molecular Formula
C20H23N3O3
Shipping Conditions
Room Temperature
Storage Conditions
At least 6 months at -20°C.
Calculated Molecular Weight
353.4 Da

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Alternative Products

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MBS131573BI-9564 (BI 9564; BI9564)
MBS3602927-01BI-9564
442674-01BI 9564
A16196-25BI-9564 25mg
A16196-50BI-9564 50mg
A16196-5BI-9564 5mg
A16196-100BI-9564 100mg
A16196-10BI-9564 10mg
HY-100352RBI-9564 (Standard)

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