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Metrenperone

CAT: 0804-HY-121311Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-121311Size:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Metrenperone is an inhibitor for 5-HT2 receptor. Metrenperone exhibits α1 and α2 antagonist activity as well as anti-H1 and anti-dopaminergic efficacy. Metrenperone can lower the blood pressure, enhances bradycardia in peripheral ischemia, inhibits serotonin-induced platelet aggregation, and antagonizes serotonin-mediated vasoconstriction. Metrenperone promotes the repair of acutely damaged collagen tissue[1][2].
CAS Number
81043-56-3
UNSPSC
12352005
Target
Adrenergic Receptor; Serotonin Transporter
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/metrenperone.html
Smiles
O=C1C(CCN2CCC(CC2)C(C3=CC=C(C=C3)F)=O)=C(N=C4N1C=C(C=C4)C)C
Molecular Formula
C24H26FN3O2
Molecular Weight
407.48
References & Citations
[1]Oryan A, et al., Effects of a serotonin S2-receptor blocker on healing of acute and chronic tendon injuries. J Invest Surg. 2009 Jul-Aug;22 (4) :246-55.|[2]Linden A, et al., Cardiovascular response to intravenous administration of 5-hydroxytryptamine after type-2 receptor blockade, by metrenperone, in healthy calves. Vet J. 1999 Jan;157 (1) :31-7.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
Launched
Isoform
α adrenergic receptor

Alternative Products

CatalogName
GTR19198877-01Metrenperone
sc-484554Metrenperone-d4

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