Products for Research Use Only

PKRA83 hydrochloride

CAT: 0013-GTR19264597-01Size: 50 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19264597-01Size:50 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
PKRA83 (PKRA7) hydrochloride is a potent prokinetic (PK2) antagonist capable of crossing the blood-brain barrier, competitively inhibiting PK2 from binding to its receptors PKR1 and PKR2. It effectively suppresses PK2 receptors, with IC50 values of 5.0 nM for PKR1 and 8.2 nM for PKR2, and exhibits anticancer, anti-arthritis, and anti-angiogenic activities.
Storage Conditions
-20°C
Notes
For research use only.

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