Products for Research Use Only

RSK-IN-2

CAT: 0013-GTR19258304-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19258304-01Size:10 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
RSK-IN-2 (Compound 3e) is an inhibitor of RSK, showing IC50 values of 37.89 nM for RSK2, 30.78 nM for RSK1, 20.51 nM for RSK3, and 91.28 nM for RSK4. It suppresses tumor cell proliferation, induces apoptosis, and causes cell cycle arrest at the G2/M phase.
CAS Number
3011713-80-4
Field of Research
Cell Biology, Signal Transduction
Smiles
O=C (NCCO) C=1C=CC=CC1NC2=NC (=NC=C2Cl) NC3=CC=C (C=C3OC) N4CCN (C) CC4
Molecular Formula
C25H30ClN7O3
Molecular Weight
512.004
Storage Conditions
-20°C
Notes
For research use only.