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TRPV1 antagonist 11

CAT: 0013-GTR19258301-01Size: 25 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19258301-01Size:25 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
TRPV1 antagonist 11 (compound 2ac) is a highly potent TRPV1 antagonist with an IC50 of 29.3 nM. It also acts as a μ-opioid receptor (MOR) agonist with a Ki of 60.3 nM. This pyrimidinylpiperazine compound provides analgesic effects by antagonizing TRPV1 and activating MOR. In mouse models of formalin-induced pain, TRPV1 antagonist 11 demonstrates effective dose-dependent antinociceptive properties.
Field of Research
Metabolism Research, Neuroscience, Neuroscience; Pharmacology & Drug Discovery, Pharmacology & Drug Discovery
Molecular Formula
C31H37N7O2
Storage Conditions
-20°C
Notes
For research use only.

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