Products for Research Use Only

DA-0157

CAT: 0013-GTR19250534-01Size: 50 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19250534-01Size:50 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
DA-0157 is a dual EGFR/ALK inhibitor designed to combat resistance mutations in NSCLC, showing potent in vitro activity against models like EGFR Del19/T790M/C797S and ALK-L1196M. It demonstrates oral bioavailability and antitumor efficacy in mouse models, supporting its use in preclinical oncology research.
CAS Number
2756978-82-0
Field of Research
Cardiovascular Research, Metabolism Research, Signal Transduction
Smiles
O=P (C1=CC (=CC=C1NC2=NC (=NC=C2Br) NC=3C=C (C (=CC3OC) N4CCC (N5CCN (C) CC5) CC4) C) C) (C) C
Molecular Formula
C31H43BrN7O2P
Molecular Weight
656.597
Storage Conditions
-20°C
Notes
For research use only.

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