Products for Research Use Only

STX-478

CAT: 0013-GTR19231151-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19231151-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
STX-478 is a brain-penetrant, selective PI3Kα inhibitor for research use. It demonstrates anticancer activity in preclinical models, inhibiting tumor growth in studies relevant to breast cancer and other solid tumors.
CAS Number
2883540-92-7
Product Name Alternative
PI3Kα
Field of Research
Signal Transduction
Purity
98.31% (May vary between batches)
Solubility
DMSO:100 mg/mL (249.2 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:5 mg/mL (12.46 mM)
Smiles
[C@H] (NC (NC=1C=NC (N) =NC1) =O) (C (F) (F) F) C2=C (C) C=3C (O2) =C (F) C=C (F) C3
Molecular Formula
C16H12F5N5O2
Molecular Weight
401.29
Storage Conditions
-20°C
Notes
For research use only.