Products for Research Use Only

Difelikefalin HCl

CAT: 0013-GTR19210481-01Size: 100 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19210481-01Size:100 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Difelikefalin HCl is a potent and selective κ-opioid receptor (KOR) agonist, as demonstrated by its low-nanomolar EC50 in cellular assays. It exhibits in vivo efficacy, reducing pain-related writhing and KOR antagonist-induced scratching in mice. This compound is a valuable research tool for studying KOR pharmacology in neurobiology, pruritus, and pain research contexts.
CAS Number
2711717-77-8
Smiles
C ([C@H] (NC ([C@H] (NC ([C@@H] (CC1=CC=CC=C1) NC ([C@@H] (CC2=CC=CC=C2) N) =O) =O) CC (C) C) =O) CCCCN) (=O) N3CCC (C (O) =O) (N) CC3.Cl
Molecular Formula
C36H53N7O6.xHCl
Molecular Weight
789.237
Storage Conditions
-20°C
Notes
For research use only.