Products for Research Use Only

MZP-54

CAT: 0013-GTR19204274-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19204274-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
MZP-54 is a PROTAC molecule that selectively degrades BRD3 and BRD4 proteins, exhibiting high affinity for the BRD4 BD2 domain with a Kd of 4 nM. It serves as a chemical probe for studying BET protein function in oncology and transcriptional regulation research, applicable in both cellular and in vivo models.
CAS Number
2010159-47-2
Field of Research
Epigenetics & Chromatin, Pharmacology & Drug Discovery
Smiles
N ([C@H]1C=2C (N (C (C) =O) [C@@H] (C) C1) =CC=C (C2) C3=CC=C (C (NCCOCCOCCOCC (N[C@H] (C (=O) N4[C@H] (C (NCC5=CC=C (C=C5) C=6SC=NC6C) =O) C[C@@H] (O) C4) [C@@] (C) (C) C) =O) =O) C=C3) C7=CC=C (Cl) C=C7
Molecular Formula
C55H66ClN7O9S
Molecular Weight
1036.67
Storage Conditions
-20°C
Notes
For research use only.