Products for Research Use Only

Sigma-LIGAND-1

CAT: 0013-GTR19204466-01Size: 1 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0013-GTR19204466-01Size:1 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
Sigma-LIGAND-1 is a selective sigma receptor ligand exhibiting high affinity at the DTG and PPP binding sites, with IC50 values of 16 nM and 19 nM, respectively. It shows significantly lower affinity for the dopamine D2 receptor (Ki = 4000 nM) . This profile makes it a useful research tool for investigating sigma receptor function in neuropharmacological studies, both in vitro and in vivo.
CAS Number
139652-01-0
Product Name Alternative
DTG site of sigma receptor, PPP site of sigma receptor, Sigma LIGAND 1, Sigma receptor, SigmaLIGAND1, Sigma-LIGAND-1, Sigmareceptor, σ-LIGAND-1
Field of Research
Pharmacology & Drug Discovery
Purity
99.89% (May vary between batches)
Solubility
DMSO:90 mg/mL (206.63 mM)
Smiles
Cc1c (oc2ccc (OCCCCCCN3CCC (O) CC3) cc2c1=O) -c1ccccc1
Molecular Formula
C27H33NO4
Molecular Weight
435.56
Storage Conditions
-20°C
Notes
For research use only.