Products for Research Use Only

EGFR/HER2-IN-4

CAT: 0013-GTR19184458-01Size: 25 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19184458-01Size:25 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
EGFR/HER2-IN-4 is an orally bioavailable, irreversible dual inhibitor of EGFR, effective against mutant forms including L858R/T790M (IC50: 0.6 nM) . It demonstrates potent kinase inhibition in vitro and significant anti-tumor efficacy in vivo, making it a valuable chemical probe for non-small cell lung cancer research.
Field of Research
Cardiovascular Research, Cell Biology, Signal Transduction
Storage Conditions
-20°C
Notes
For research use only.