Products for Research Use Only

MDR-652

CAT: 0013-GTR19172771-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19172771-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
MDR-652 is a potent, nonpungent TRPV1 agonist with high affinity (Ki: 11.4 nM hTRPV1) and functional potency (EC50: 5.05 nM hTRPV1) . Its strong topical analgesic properties support research in pain pathways, inflammation, and neurobiology, applicable in both in vitro receptor studies and in vivo models of nociception.
CAS Number
1933528-96-1
Product Name Alternative
Activity, analgesic, MDR 652, MDR652, MDR-652, hTRPV1, ligand, Inhibitor, inhibit, pain, neuropathic, Transient receptor potential channels, TRP Channel, TRPChannel, TRPV Channel, TRPV1, TRPVChannel
Field of Research
Pharmacology & Drug Discovery
Purity
95.04% (May vary between batches)
Solubility
10% DMSO+40% PEG300+5% Tween 80+45% Saline:5 mg/mL (11.16 mM) ; DMSO:249 mg/mL (555.87 mM)
Smiles
CC (C) (C) c1nc (c (CNC (=O) Nc2ccc (CO) c (F) c2) s1) -c1cccc (Cl) c1
Molecular Formula
C22H23ClFN3O2S
Molecular Weight
447.95
Storage Conditions
-20°C
Notes
For research use only.

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