Products for Research Use Only

Samelisant

CAT: 0013-GTR19166773-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19166773-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Samelisant (SUVN-G3031) is a potent, selective inverse agonist of the histamine H3 receptor, exhibiting Kis of 8.7 nM (human) and 9.8 nM (rat) . It demonstrates anticataplectic activity in vivo and is a valuable research tool for investigating narcolepsy and related sleep/wake disorders in both in vitro and in vivo experimental models.
CAS Number
1394808-82-2
Product Name Alternative
H3 receptor, Histamine Receptor, HistamineReceptor, SUVN-G 3031, SUVN-G3031, SUVN-G-3031, Samelisant
Field of Research
Immunology & Inflammation, Neuroscience, Pharmacology & Drug Discovery
Purity
99.09% (May vary between batches)
Solubility
DMSO:50 mg/mL (133.87 mM)
Smiles
O (C1CCN (CC1) C2CCC2) C3=CC=C (NC (CN4CCOCC4) =O) C=C3
Molecular Formula
C21H31N3O3
Molecular Weight
373.49
Storage Conditions
-20°C
Notes
For research use only.