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PF-CBP1

CAT: 0013-GTR19162896-06Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19162896-06Size:10 mg
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Description
A potent, highly selective CBP/p300 bromodomains inhibitor with IC50 of 125 nM and 363 nM, respectively; displays >100-fold selectivity for the bromodomain of CBP over those of BRD4 and a panel of other proteins; reduces the expression of inflammatory cytokines by LPS-stimulated primary macrophages, also suppresses the expression of RGS4 in primary cortical neurons.
CAS Number
1962928-21-7
Product Name Alternative
PF CBP1
Field of Research
Cell Biology
Purity
>98% (HPLC)
Solubility
DMSO: 100 mg/mL (< 1 mg/ml refers to the product slightly soluble or insoluble)
Smiles
CCCOC1=CC=C (C=C1) CCC2=NC3=C (N2CCN4CCOCC4) C=CC (=C3) C5=C (ON=C5C) C
Molecular Formula
C29H36N4O3
Molecular Weight
488.6
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Other Product Names
4- (2- (5- (3,5-dimethylisoxazol-4-yl) -2- (4-propoxyphenethyl) -1H-benzo[d]imidazol-1-yl) ethyl) morpholine

Chemical Information

PF-Cbp1
CAS Number1962928-21-7
PubChem CID119081417
IUPAC Name4-[2-[5-(3,5-dimethyl-1,2-oxazol-4-yl)-2-[2-(4-propoxyphenyl)ethyl]benzimidazol-1-yl]ethyl]morpholine
Molecular FormulaC29H36N4O3
Molecular Weight488.6
XLogP5
Topological Polar Surface Area65.6
Hydrogen Bond Donor Count0
Hydrogen Bond Acceptor Count6
Rotatable Bond Count10
Heavy Atom Count36
Formal Charge0
Complexity654
SMILES
CCCOC1=CC=C(C=C1)CCC2=NC3=C(N2CCN4CCOCC4)C=CC(=C3)C5=C(ON=C5C)C
InChI
InChI=1S/C29H36N4O3/c1-4-17-35-25-9-5-23(6-10-25)7-12-28-30-26-20-24(29-21(2)31-36-22(29)3)8-11-27(26)33(28)14-13-32-15-18-34-19-16-32/h5-6,8-11,20H,4,7,12-19H2,1-3H3
InChIKey
CGWBJJZOKGZCSJ-UHFFFAOYSA-N
Chemical Structure
2D Structure
2D structure of PF-Cbp1
CAS: 1962928-21-7
CID: 119081417
Formula: C29H36N4O3
MW: 488.6
Interactive 3D Structure
Loading 3D structure...
View on PubChemRaw 3D data
Computed Properties
PropertyValue
Molecular Weight488.6
XLogP35
Hydrogen Bond Donor Count0
Hydrogen Bond Acceptor Count6
Rotatable Bond Count10
Exact Mass488.27874102
Monoisotopic Mass488.27874102
Topological Polar Surface Area65.6 Ų
Heavy Atom Count36
Formal Charge0
Complexity654
Isotope Atom Count0
Defined Atom Stereocenter Count0
Undefined Atom Stereocenter Count0
Defined Bond Stereocenter Count0
Undefined Bond Stereocenter Count0
Covalently-Bonded Unit Count1
Compound Is CanonicalizedYes

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