Abarelix

CAT: 0013-GTR19155656-01Size: 200 mgDry Ice: NoHazardous: No

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CAT#:0013-GTR19155656-01Size:200 mg

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Description

Abarelix is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment. (In Vitro) :Abarelix (30 and 300 μg/mL) causes significantly increased histamine release. Abarelix is the first GnRH antagonist to be developed, and can produce rapid and sustained decreases in testosterone to castrate levels without the need for co-administration of an antiandrogen, and with a very low complication rate in the short term. Abarelix demonstrates to promptly and substantially reduce follicle-stimulating hormone levels to lower than LHRH agonist. Abarelix does not cause a surge in serum testosterone that can precipitate a flare phenomenon or worsening of disease, particularly dangerous for patients with metastatic, symptomatic disease, and produces medical castration more quickly.

CAS Number

183552-38-7

Product Name Alternative

R3827 | PPI 149

Field of Research

Pharmacology & Drug Discovery

Purity

>98% (HPLC)

Solubility

DMSO:14.2 mg/mL (10.03 mM)

Smiles

C[C@H] (C (=O) N) NC (=O) [C@@H]1CCCN1C (=O) [C@H] (CCCCNC (C) C) NC (=O) [C@H] (CC (C) C) NC (=O) [C@@H] (CC (=O) N) NC (=O) [C@H] (CC2=CC=C (C=C2) O) N (C) C (=O) [C@H] (CO) NC (=O) [C@@H] (CC3=CN=CC=C3) NC (=O) [C@@H] (CC4=CC=C (C=C4) Cl) NC (=O) [C@@H] (CC5=CC6=CC=CC=C6C=C5) NC (=O) C

Molecular Formula

C72H95ClN14O14

Molecular Weight

1416.06

Storage Conditions

Storage temperature: -20°C. Stability: ≥ 2 years

Notes

For research use only.

Alternative Products

Catalog	Name
BA5366-5	Abarelix
T68701-01	Abarelix acetate
KGB80417-01	Abarelix (acetate)

Abarelix

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