BRD9 Degrader-2
CAT:
804-HY-163809
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- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No

BRD9 Degrader-2
- CAS Number: 3033018-68-4
- UNSPSC Description: BRD9 Degrader-2 (Compound B11) is a BRD9 degrader (DC50 ≤1.25 nM; Dmax≥75%). BRD9 Degrader-2 can be used for research of cancers[1].
- Target Antigen: E1/E2/E3 Enzyme; Epigenetic Reader Domain; Molecular Glues
- Type: Reference compound
- Related Pathways: Epigenetics;Metabolic Enzyme/Protease;PROTAC
- Applications: Cancer-programmed cell death
- Field of Research: Cancer
- Assay Protocol: https://www.medchemexpress.com/brd9-degrader-2.html
- Smiles: N#C/C(C(N1CCC2=C(C1C)C=CC=C2CN3CCN(CC3)CC4=C(OC)C=C(C5=CN(C)C(C(C)=C5C)=O)C=C4OC)=O)=C\C6=NC(C(F)(F)F)=CS6
- Molecular Weight: 760.87
- References & Citations: [1]David MCGARRY, et al. Compounds for targeted protein degradation. Patent. WO2024057021A1
- Shipping Conditions: Room temperature
- Clinical Information: No Development Reported