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Goxalapladib

CAT: 0804-HY-169114-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-169114-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Goxalapladib is a 5-HT6 receptor modulator that blocks lipoprotein-associated phospholipase A2 (Lp-PLA2) activity. Goxalapladib is promising for research of atherosclerosis-associated cardiovascular diseases[1].
CAS Number
412950-27-7
UNSPSC
12352005
Target
5-HT Receptor; Phospholipase
Type
Reference compound
Related Pathways
GPCR/G Protein; Metabolic Enzyme/Protease; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/goxalapladib.html
Smiles
O=C1C=C(CCC2=C(F)C(F)=CC=C2)N(CC(N(C3CCN(CC3)CCOC)CC4=CC=C(C5=CC=C(C(F)(F)F)C=C5)C=C4)=O)C6=NC=CC=C16
Molecular Formula
C40H39F5N4O3
Molecular Weight
718.75
References & Citations
[1]Feuerstein GZ, et al. Discontinued drugs in 2006: cardiovascular drugs translational medicine perspective. Expert Opin Investig Drugs. 2007 Sep;16 (9) :1315-26.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
Phase 1
Isoform
5-HT6 Receptor; MUC2

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CatalogName
T67799-01Goxalapladib

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