Sarafotoxin S6c

• Target:

  Endothelin Receptor

• Related Pathways:

  GPCR/G Protein

• Bioactivity:

  Highly selective ETB endothelin receptor agonist (Ki values are 0.29 and 28000 nM at ETB and ETA receptors respectively) .

• Smiles:

  C ([C@H] (NC ([C@@H] (NC ([C@@H] (NC ([C@@H] (NC ([C@@H] (NC ([C@H] (CC1=CN=CN1) NC (=O) [C@H]2NC (=O) [C@H] (CC3=CC=CC=C3) NC (=O) [C@H] (CC (N) =O) NC (=O) [C@H] (CC (C) C) NC (=O) [C@]4 (NC (=O) [C@H] (CCC (O) =O) NC (=O) [C@H] (CCC (O) =O) NC (=O) [C@H] (CC (O) =O) NC (=O) [C@] ([C@@H] (C) O) (NC (=O) [C@H] (CCSC) NC (=O) [C@H] (CC (O) =O) NC (=O) [C@H] (CC (N) =O) NC (=O) [C@@] (NC (=O) [C@] ([C@@H] (C) O) (NC (=O) [C@@H] (N) CSSC2) [H]) (CSSC4) [H]) [H]) [H]) =O) CCC (N) =O) =O) CC (O) =O) =O) [C@@H] (C) C) =O) [C@H] (CC) C) =O) C (O) =O) C=5C=6C (NC5) =CC=CC6

• Molecular Formula:

  C103H147N27O37S5

• Molecular Weight:

  2516

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  121695-87-2