Products for Research Use Only

AdTx1

CAT: 0931-TP2086Size: 1 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0931-TP2086Size:1 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Target
Adrenergic Receptor
Related Pathways
Neuroscience, GPCR/G Protein
Bioactivity
Selective, high affinity, non-competitive α1A adrenoceptor antagonist (Ki = 0.35 nM) . Exhibits no significant activity against a range of other GPCRs, including α2A, β1 and β2 adrenoceptors. Antagonizes effects of phenylephrine on isolated rabbit prostate muscle in vitro and on intra-urethral pressure in rats.
Molecular Formula
C310H481N87O100S8
Molecular Weight
7283.22
Shipping Conditions
Ice Packs
Storage Temperature
-20°C