GR 64349

• Target :

  Neurokinin receptor

• Related Pathways :

  Neuroscience|||GPCR/G Protein

• Bioactivity :

  Potent and selective tachykinin NK2 receptor agonist (EC50 = 3.7 nM in rat colon) . Displays > 1000- and > 300-fold selectivity over NK1 and NK3 receptors respectively. Active in vivo.

• Smiles :

  CSCC[C@H](NC(=O)[C@H](CC(C)C)N1CC[C@@H](NC(=O)[C@@H](NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](CO)NC(=O)[C@H](CC(O)=O)NC(=O)[C@@H](N)CCCCN)C(C)C)C1=O)C(N)=O

• Molecular Formula :

  C42H68N10O11S

• Molecular Weight :

  921.12

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  137593-52-3