γ1-MSH

CAT: 0931-TP1892Size: 1 mgDry Ice: NoHazardous: No
CAT#:0931-TP1892Size:1 mg
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AVAILABILITY
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
72629-65-3
Target
Melanocortin Receptor
Related Pathways
Neuroscience|||GPCR/G Protein
Bioactivity
Endogenous melanocortin MC3 receptor agonist (pKi = 7.46) that displays ~ 40-fold selectivity over MC4. Increases the release of extracellular dopamine, which induces grooming and vertical activity (rearing) in rats. Exhibits hypertensive, tachycardic and short-term analgesic activity in vivo.
Smiles
C([C@H](NC([C@@H](NC([C@H](CC1=CC=CC=C1)NC([C@H](CC2=CN=CN2)NC(CNC([C@@H](NC([C@@H](NC([C@H](CC3=CC=C(O)C=C3)N)=O)[C@@H](C)C)=O)CCSC)=O)=O)=O)=O)CCCNC(=N)N)=O)C(N[C@H](C(N[C@H](C(N[C@@H](CC4=CC=CC=C4)C(N)=O)=O)CCCNC(=N)N)=O)CC(O)=O)=O)C=5C=6C(NC5)=CC=CC6
Molecular Formula
C72H97N21O14S
Molecular Weight
1512.76
Shipping Conditions
Cool pack
Storage Temperature
-20°C