CL 218872
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


CL 218872
Target :
GABA ReceptorRelated Pathways :
Neuroscience|||Membrane transporter/Ion channelPurity :
0.9997Bioactivity :
CL 218872 is a benzodiazepine agonist displaying selectivity for ?1 subunit-containing GABAA receptors (Ki values are 130, 1820, 1530, > 10000, 490 and > 10000 nM for ?1, ?2, ?3, ?4, ?5 and ?6-subunit containing receptors respectively) . Orally active anxiolytic and anticonvulsant in vivo.Smiles :
CC=1N2C(C=CC(=N2)C3=CC(C(F)(F)F)=CC=C3)=NN1Molecular Formula :
C13H9F3N4Molecular Weight :
278.23Shipping Conditions :
Cool packStorage Temperature :
-20°CCAS Number :
66548-69-4

