TC-I2000
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


TC-I2000
Target:
TRP/TRPV ChannelRelated Pathways:
Membrane transporter/Ion channelPurity:
0.9978Bioactivity:
TC-I2000 is an TRPM8 channel blocker. Inhibits icilin-induced TRPM8 channel activation in rTRPM8-expressing CHO cells with IC50 of 53 nM.Smiles:
C(NC1=CC=C(F)C=C1)(=O)N2C(C=3C(CC2)=CC=CC3)C4=CC=C(C(F)(F)F)C=C4Molecular Formula:
C23H18F4N2OMolecular Weight:
414.4Shipping Conditions:
Cool packStorage Temperature:
-20°CCAS Number:
1159996-20-9
