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Nelotanserin

CAT: 0931-T7350-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0931-T7350-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
839713-36-9
Target
5-HT Receptor
Related Pathways
Neuroscience, GPCR/G Protein
Purity
0.9988
Bioactivity
Nelotanserin (APD125) is a potent 5-HT2A inverse agonist (IC50 : 1.7 nM), a moderately potent 5-HT2C partial inverse agonist t (IC50 :79 nM) and a weak 5-HT2B inverse agonistt (IC50 : 791 nM) .
Smiles
COc1ccc(NC(=O)Nc2ccc(F)cc2F)cc1-c1c(Br)cnn1C
Molecular Formula
C18H15BrF2N4O2
Molecular Weight
437.24
Shipping Conditions
Ice Packs
Storage Temperature
-20°C