CPI-360

• Target:

  Histone Methyltransferase|||Apoptosis

• Related Pathways:

  Apoptosis|||Chromatin/Epigenetic

• Purity:

  0.9989

• Bioactivity:

  CPI-360 is a small molecule EZH2 inhibitor (IC50: 0.002 ?M, EC50: 0.080 ?M) that shows antitumor activity in an EZH200-dependent tumor xenograft model.

• Smiles:

  [C@H](C)(N1C=2C(C(C(NCC3=C(OC)C=C(C)NC3=O)=O)=C1C)=CC=CC2)C4CCOCC4

• Molecular Formula:

  C25H31N3O4

• Molecular Weight:

  437.53

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  1802175-06-9