Products for Research Use Only

GKA50 quarterhydrate

CAT: 0931-T63019-01Size: 25 mgDry Ice: NoHazardous: No
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CAT#:0931-T63019-01Size:25 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
Others, Glucokinase
Related Pathways
Metabolism, Others
Bioactivity
GKA50 quarterhydrate is a potent glucokinase activator with an EC50 value of 33 nM. This glucose-like activator of β-cell metabolism in rodent and human pancreatic islets is a Ca2+-dependent regulator of insulin secretion. It stimulates insulin secretion in mouse islets and significantly reduces blood glucose in high-fat-fed female rats.
Molecular Formula
C26H30N2O7
Molecular Weight
469.01
Shipping Conditions
Ice Packs
Storage Temperature
-20°C