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CPI-1612

CAT: 0931-T62721-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T62721-01Size:10 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2374971-81-8
Target
Others, Histone Acetyltransferase
Related Pathways
Others, Chromatin/Epigenetic
Bioactivity
CPI-1612 is a potent, orally active EP300/CBP histone acetyltransferase (HAT) inhibitor that acts on EP300 HAT (IC50: 8.1 nM) . CPI-1612 exhibits anticancer effects.
Smiles
C[C@H](CN[C@@H](C(=O)Nc1ccc(cn1)-c1cnn(C)c1)c1ccccc1)c1ccc(cc1)C#N
Molecular Formula
C27H26N6O
Molecular Weight
450.53
Shipping Conditions
Ice Packs
Storage Temperature
-20°C