CPI-1612

• Target:

  Others|||Histone Acetyltransferase

• Related Pathways:

  Others|||Chromatin/Epigenetic

• Bioactivity:

  CPI-1612 is a potent, orally active EP300/CBP histone acetyltransferase (HAT) inhibitor that acts on EP300 HAT (IC50: 8.1 nM) . CPI-1612 exhibits anticancer effects.

• Smiles:

  C[C@H](CN[C@@H](C(=O)Nc1ccc(cn1)-c1cnn(C)c1)c1ccccc1)c1ccc(cc1)C#N

• Molecular Formula:

  C27H26N6O

• Molecular Weight:

  450.53

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  2374971-81-8