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Camonsertib

CAT: 0931-T62083-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0931-T62083-01Size:1 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2417489-10-0
Target
ATM/ATR, mTOR
Related Pathways
DNA Damage/DNA Repair, PI3K/Akt/mTOR signaling
Purity
0.9993
Bioactivity
Camonsertib (RP-3500) is a novel, potent and selective ATR kinase inhibitor (ATRi) that exhibits potent antitumor effects with an IC50: 1.00 nM in biochemical assays.RP-3500 is 30-fold more selective for ATR than mTOR (IC50: 120 nM) and more than 2,000-fold more potent than ATM, DNA-PK and PI3Kα kinases. RP-3500 is 30 times more selective for ATR than mTOR (IC50: 120 nM), and 2,000 times more selective than ATM, DNA-PK and PI3Kα kinases.
Smiles
C[C@@H]1COCCN1c1cc(c2cnn(-c3cc[nH]n3)c2n1)[C@@]1(O)C[C@@H]2CC[C@H](C1)O2
Molecular Formula
C21H26N6O3
Molecular Weight
410.47
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

Alternative Products

CatalogName
M35617-01Camonsertib
A21870-50Camonsertib 50mg
A21870-25Camonsertib 25mg
A21870-10Camonsertib 10mg
A21870-5Camonsertib 5mg
A21870-100Camonsertib 100mg
A21870-1Camonsertib 1mg
E1108-01Camonsertib (RP-3500)
A21870-10mM-DCamonsertib 10mM * 1mL in DMSO

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