BI 2536
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


BI 2536
Target:
Apoptosis|||Epigenetic Reader Domain|||PLKRelated Pathways:
Apoptosis|||Cell Cycle/Checkpoint|||Chromatin/EpigeneticPurity:
0.9988Bioactivity:
BI2536 is an effective Plk1 inhibitor (IC50: 0.83 nM) . It has 4- and 11-fold greater selectivity than Plk2 and Plk3.Smiles:
C(C)[C@H]1N(C=2C(N(C)C1=O)=CN=C(NC3=C(OC)C=C(C(NC4CCN(C)CC4)=O)C=C3)N2)C5CCCC5Molecular Formula:
C28H39N7O3Molecular Weight:
521.65Shipping Conditions:
Cool packStorage Temperature:
-20°CCAS Number:
755038-02-9
