VPC-13789

CAT: 0931-T61653-01Size: 25 mgDry Ice: NoHazardous: No
CAT#:0931-T61653-01Size:25 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2761146-51-2
Target
Others|||Androgen Receptor
Related Pathways
Endocrinology/Hormones|||Others
Bioactivity
VPC-13789 is a highly potent, selective, and orally bioavailable antiandrogen compound that shows promise for studying and developing therapeutics for castration-resistant prostate cancer (CRPC) . In LNCaP cells, VPC-13789 effectively inhibits the transcriptional activity of the androgen receptor (AR) with an IC50 value of 0.19 ?M [1].
Smiles
FC1=C2C(C(=CN2)C3=NC4=C(C=C3)C(C(NC(C)C)=O)=CC=C4)=CC(F)=C1F
Molecular Formula
C21H16F3N3O
Molecular Weight
383.37
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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