VPC-13566

• Target:

  Androgen Receptor

• Related Pathways:

  Endocrinology/Hormones

• Purity:

  0.9955

• Bioactivity:

  VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the BF3 pocket. VPC-13566 inhibits the growth of various prostate cancer cell lines and reduces the growth of AR-dependent prostate cancer xenograft tumors in mice.

• Smiles:

  CC1=C2C (C (=CN2) C3=NC4=C (C=C3) C=CC=C4) =CC=C1

• Molecular Formula:

  C18H14N2

• Molecular Weight:

  258.32

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  218464-59-6