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H3R antagonist 2

CAT: 0931-T61603-01Size: 25 mgDry Ice: NoHazardous: No
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CAT#:0931-T61603-01Size:25 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Target
Others, Monoamine Oxidase, Histamine Receptor, Cholinesterase (ChE)
Related Pathways
Immunology/Inflammation, Others, Neuroscience, GPCR/G Protein
Bioactivity
H3R antagonist 2 (Compound 23) is a multitarget histamine H3 receptor antagonist with inhibitory effects on acetylcholinesterase, butyrylcholinesterase, and human monoamine oxidase B (hMAO B) with IC50 values of 180 nM, 880 nM, and 775 nM, respectively. With a Ki of 170 nM for hH3R, it demonstrates favorable anti-neuropathic pain and memory-enhancing effects and can cross the blood-brain barrier (BBB) [1].
Molecular Formula
C24H29NO3
Molecular Weight
379.49
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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