Products for Research Use Only

Haspin-IN-1

CAT: 0931-T60477-01Size: 25 mgDry Ice: NoHazardous: No
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CAT#:0931-T60477-01Size:25 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
Others, DYRK, Haspin Kinase, CDK
Related Pathways
Tyrosine Kinase/Adaptors, Others, Cell Cycle/Checkpoint
Bioactivity
Haspin-IN-1 (compound 2a) is an inhibitor of haspin (haploid germ cell-specific nuclear protein kinase) with an IC50 of 119 nM. It also inhibits CLK1, DYRK1A, and CDK9 with IC50 values of 221 nM, 916.3 nM, and 406.8 nM, respectively. Haspin-IN-1 has potential for developing new anticancer drugs [1].
Molecular Formula
C12H8N4O2S
Molecular Weight
272.28
Shipping Conditions
Ice Packs
Storage Temperature
-20°C