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PBRM1-BD2-IN-8

CAT: 0931-T60157-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0931-T60157-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2819989-75-6
Target
Epigenetic Reader Domain
Related Pathways
Chromatin/Epigenetic
Purity
0.9989
Bioactivity
PBRM1-BD2-IN-8 (compound 34) is a potent PBRM1 Bromodomain inhibitor with PBRM1-BD2 Kd of 4.4 μM, PBRM1-BD2 IC50 of 0.16 μM, and PBRM1-BD5 Kd of 25 μM; PBRM1-BD2-IN-8 shows anti-cancer activity.
Smiles
O=C1C=2C(NC(N1)C3=CC(C)=CC=C3)=CC=CC2Br
Molecular Formula
C15H13BrN2O
Molecular Weight
317.18
Shipping Conditions
Ice Packs
Storage Temperature
-20°C