NSC 694621

• Target:

  Epigenetic Reader Domain|||Histone Acetyltransferase

• Related Pathways:

  Chromatin/Epigenetic

• Purity:

  0.997

• Bioactivity:

  NSC 694621 is a PCAF and histone acetyltransferase (HAT) inhibitor that forms a covalent bond with Cys574, the active site of PCAF, thereby irreversibly inhibiting its acetyltransferase activity, and is able to inhibit the proliferation of SK-N-SH and HCT116 cells, which has anticancer potential.

• Smiles:

  O=C1C2=CC=CN=C2SN1C3=CC=C(OC)C=C3

• Molecular Formula:

  C13H10N2O2S

• Molecular Weight:

  258.3

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  104857-29-6