Cis-22a

• Target :

  Calcium Channel|||TRP/TRPV Channel

• Related Pathways :

  Membrane transporter/Ion channel|||Metabolism

• Purity :

  0.9999

• Bioactivity :

  Cis-22a is a TRPV6 inhibitor (IC50 = 0.32 ?M), which exhibits selectivity against related TRPV channels and calcium channels. cis-22a displays antiproliferative effects on T47D human breast cancer cells.

• Smiles :

  C(C(O)=O)(F)(F)F.CC=1C=C([C@H]2CC[C@H](CC2)N3CCN(CC3)C=4C=CC=NC4)C=CC1

• Molecular Formula :

  C24H30F3N3O2

• Molecular Weight :

  449.51

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  1819366-84-1