Bilaid C

CAT: 0931-MF-0036593-01Size: 1 mgDry Ice: NoHazardous: No
CAT#:0931-MF-0036593-01Size:1 mg
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CAS Number
2393866-13-0
Target
Opioid Receptor
Related Pathways
Neuroscience|||Endocrinology/Hormones|||GPCR/G Protein
Bioactivity
Bilaid C is a tetrapeptide ?-opioid receptor agonist (Ki= 210 nM in HEK293 cell membranes expressing the human receptor) that has been found inPenicillium.1It inhibits forskolin-induced cAMP accumulation by 77% in HEK293 cells expressing the human ?-opioid receptor when used at a concentration of 10 ?M. Bilaid C induces inward rectifying potassium channel (Kir) currents in rat locus coeruleus slices that endogenously express high levels of the ?-opioid receptor (EC50= 4.2 ?M) .
Smiles
CC(C)[C@H](NC(=O)[C@H](NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(C)C)C(=O)N[C@H](Cc1ccccc1)C(O)=O
Molecular Formula
C28H38N4O6
Molecular Weight
526.62
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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