Ecopipam

• Target:

  5-HT Receptor|||Dopamine Receptor|||Adrenergic Receptor

• Related Pathways:

  GPCR/G Protein|||Neuroscience

• Purity:

  0.9968

• Bioactivity:

  Ecopipam (UNII-0X748O646K) is a potent, selective, and orally active antagonist of dopamine D1/D5 receptors, with Kis of 1.2 nM and 2.0 nM, respectively. Ecopipam demonstrates more than 40-fold selectivity over D2, D4, 5-HT, and ?2a receptors (Ki=0.98, 5.52, 0.08, and 0.73 ?M, respectively) . It is used in research on schizophrenia and obesity.

• Smiles:

  CN1[C@@]2([C@@](C=3C(=CC(Cl)=C(O)C3)CC1)(C=4C(CC2)=CC=CC4)[H])[H]

• Molecular Formula:

  C19H20ClNO

• Molecular Weight:

  313.82

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  112108-01-7