Products for Research Use Only

GS-462808

CAT: 0931-T27437-01Size: 25 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0931-T27437-01Size:25 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
CAS Number
1354198-41-6
Target
Others, Sodium Channel
Related Pathways
Others, Membrane transporter/Ion channel
Bioactivity
GS-462808 is a late sodium current inhibitor of the cardiac Nav1.5 channel. GS-462808 had lower brain penetration and serendipitously lower activity at the brain isoforms.
Smiles
O=C1N2C(=NN1CC3=NC(C)=NO3)C=CC(=C2)C4=CC=C(OC(F)(F)F)C=C4
Molecular Formula
C17H12F3N5O3
Molecular Weight
391.3
Shipping Conditions
Ice Packs
Storage Temperature
-20°C