CP 154,526

• Target :

  Others|||CRFR

• Related Pathways :

  GPCR/G Protein|||Others

• Bioactivity :

  CP 154,526 is a selective CRF1 receptor antagonist (Ki = 2.7 nM) . CP 154,526 blocks CRF-induced activation of adenylate cyclase and the HPA axis.

• Smiles :

  N(CCCC)(CC)C1=C2C(N(C=C2C)C3=C(C)C=C(C)C=C3C)=NC(C)=N1

• Molecular Formula :

  C23H32N4

• Molecular Weight :

  364.53

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  157286-86-7