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Gandotinib

CAT: 0931-T2638-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0931-T2638-01Size:5 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1229236-86-5
Target
FGFR, VEGFR, FLT, JAK
Related Pathways
Chromatin/Epigenetic, Tyrosine Kinase/Adaptors, JAK/STAT signaling, Stem Cells, Angiogenesis
Purity
0.9986
Bioactivity
LY2784544 (Gandotinib (LY2784544) ) is a potent JAK2 inhibitor (IC50: 3 nM), effective in JAK2V617F (Ki: 0.245 nM) . The selectivity is higher 8- and 20-fold than JAK1 and JAK3.
Smiles
C(C=1C=2N(C(CC3=C(F)C=C(Cl)C=C3)=C(C)N2)N=C(NC=4C=C(C)NN4)C1)N5CCOCC5
Molecular Formula
C23H25ClFN7O
Molecular Weight
469.94
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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