BX-912
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


BX-912
Target :
PKA|||PDK|||Chk|||VEGFR|||Apoptosis|||CDKRelated Pathways :
Angiogenesis|||Apoptosis|||PI3K/Akt/mTOR signaling|||Tyrosine Kinase/Adaptors|||Cell Cycle/CheckpointPurity :
0.9934Bioactivity :
BX-912 is a specific inhibitor of 3-Phosphoinositide-dependent Kinase-1 (PDK1, IC50: 12 nM) . The selectivity of BX-912 is more 10 fold than C-Kit, EGFR, PKA, PKC etc.Smiles :
Brc1cnc(Nc2cccc(NC(=O)N3CCCC3)c2)nc1NCCc1cnc[nH]1Molecular Formula :
C20H23BrN8OMolecular Weight :
471.35Shipping Conditions :
Cool packStorage Temperature :
-20°CCAS Number :
702674-56-4

