TM-N1324

• Target:

  GHSR

• Related Pathways:

  GPCR/G Protein

• Purity:

  0.9988

• Bioactivity:

  TM-N1324 is a GPR39 agonist. TM-N1324 activates human GPR39 with high efficacy and potencies of 280 nM and 9 nM in the absence and presence of Zn2+, respectively. TM-N1324 has similar potencies to murine GPR39 with EC50s of 180 nM and 5 nM, respectively.

• Smiles:

  Cc1nn(c2NC(=O)CC(c12)c1ccc(F)cc1Cl)-c1ncnc2[nH]cnc12

• Molecular Formula:

  C18H13ClFN7O

• Molecular Weight:

  397.79

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  1144477-35-9