RPR-260243
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


RPR-260243
Target :
Potassium Channel|||OthersRelated Pathways :
Others|||Membrane transporter/Ion channelBioactivity :
RPR-260243 is a novel activator of HERG and modifies HERG currents inhibited by dofetilide (IC50 = 58 nM) .Smiles :
COc1ccc2nccc(C(=O)CC[C@@H]3CCN(CC#Cc4cc(F)cc(F)c4F)C[C@@H]3C(O)=O)c2c1Molecular Formula :
C28H25F3N2O4Molecular Weight :
510.5Shipping Conditions :
Cool packStorage Temperature :
-20°CCAS Number :
668463-35-2

