RPR-260243
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


RPR-260243
Target:
Potassium Channel|||OthersRelated Pathways:
Others|||Membrane transporter/Ion channelBioactivity:
RPR-260243 is a novel activator of HERG and modifies HERG currents inhibited by dofetilide (IC50 = 58 nM) .Smiles:
COc1ccc2nccc(C(=O)CC[C@@H]3CCN(CC#Cc4cc(F)cc(F)c4F)C[C@@H]3C(O)=O)c2c1Molecular Formula:
C28H25F3N2O4Molecular Weight:
510.5Shipping Conditions:
Cool packStorage Temperature:
-20°CCAS Number:
668463-35-2
