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PCS1055 dihydrochloride

CAT: 0931-T16443-01Size: 25 mgDry Ice: NoHazardous: No
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CAT#:0931-T16443-01Size:25 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
361979-40-0
Target
Cholinesterase (ChE), AChR, Others
Related Pathways
Others, Neuroscience
Bioactivity
PCS1055 dihydrochloride is an effective, selective, and competitive muscarinic M4 receptor antagonist (IC50: 18.1 nM and a Kd: 5.72 nM) . PCS1055 dihydrochloride is also a potent AChE inhibitor (IC50 s: 22 nM and 120 nM for electric eel and human AChE, respectively) . PCS1055 dihydrochloride inhibits radioligand [3H]-NMS binding to the M4 receptor (Ki: 6.5 nM) . PCS1055 dihydrochloride shows >100-fold selectivity over M1-, M3-, and M5-receptors and 30-fold selectivity at the M2 receptor.
Smiles
C1(N=NC(NCCC2CCN(CC2)CC3=CC=CC=C3)=C4)=C4CCCC5=CC=CC=C15.Cl.Cl
Molecular Formula
C27H34Cl2N4
Molecular Weight
485.49
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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