MA-2029

• Target:

  Motilin Receptor|||Others

• Related Pathways:

  GPCR/G Protein|||Others

• Bioactivity:

  MA-2029 is selective for the motilin receptor over various other receptors and ion channels. MA-2029 is a selective and competitive motilin receptor antagonist (IC50=4.9 nM) . MA-2029 may be useful for gastrointestinal disorders associated with disturbed gastrointestinal motility.

• Smiles:

  CCNC (=O) [C@H] (Cc1ccc (O) c (c1) C (C) (C) C) NC (=O) [C@H] (C (C) C) N (C) C (=O) [C@H] (Cc1ccc (F) cc1) NC

• Molecular Formula:

  C31H45FN4O4

• Molecular Weight:

  556.71

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  287206-61-5