MA-2029

• Target :

  Motilin Receptor|||Others

• Related Pathways :

  GPCR/G Protein|||Others

• Bioactivity :

  MA-2029 is selective for the motilin receptor over various other receptors and ion channels. MA-2029 is a selective and competitive motilin receptor antagonist (IC50=4.9 nM) . MA-2029 may be useful for gastrointestinal disorders associated with disturbed gastrointestinal motility.

• Smiles :

  CCNC(=O)[C@H](Cc1ccc(O)c(c1)C(C)(C)C)NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H](Cc1ccc(F)cc1)NC

• Molecular Formula :

  C31H45FN4O4

• Molecular Weight :

  556.71

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  287206-61-5