Fenobam

• Target:

  Apoptosis|||GluR

• Related Pathways:

  Neuroscience|||Apoptosis

• Purity:

  0.9993

• Bioactivity:

  Fenobam shows inverse agonist activity which blocks the mGlu5 receptor basal activity (IC50: 84 nM) . Fenobam has anxiolytic activity. Fenobam is a selective and non-competitive mGluR5 antagonist acting at an allosteric modulatory site (Kd values are 54 and 31 nM for rat and human recombinant mGlu5 receptors, respectively) .

• Smiles:

  CN1CC (=O) N=C1NC (=O) Nc1cccc (Cl) c1

• Molecular Formula:

  C11H11ClN4O2

• Molecular Weight:

  266.68

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  57653-26-6